Mitiglinide calcium hydrate
CAS No. 207844-01-7
Mitiglinide calcium hydrate ( KAD-1229 calcium hydrate;S-21403 calcium hydrate )
Catalog No. M13230 CAS No. 207844-01-7
An insulin secretion stimulator by closing the ATP-sensitive potassium KATP channels in pancreatic β cells.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
100MG | 37 | In Stock |
|
500MG | 109 | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameMitiglinide calcium hydrate
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NoteResearch use only, not for human use.
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Brief DescriptionAn insulin secretion stimulator by closing the ATP-sensitive potassium KATP channels in pancreatic β cells.
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DescriptionAn insulin secretion stimulator by closing the ATP-sensitive potassium KATP channels in pancreatic β cells; has potent hypoglycemic effects.Diabetes Approved
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SynonymsKAD-1229 calcium hydrate;S-21403 calcium hydrate
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PathwayCell Cycle/DNA Damage
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TargetPotassium Channel
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RecptorPotassiumChannel
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Research AreaMetabolic Disease
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IndicationDiabetes
Chemical Information
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CAS Number207844-01-7
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Formula Weight353.46
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Molecular FormulaC19H25NO3 . 1/2 Ca . H2O
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESC1CC[C@H]2CN(C[C@H]2C1)C(=O)C[C@H](CC3=CC=CC=C3)C(=O)[O-].C1CC[C@H]2CN(C[C@H]2C1)C(=O)C[C@H](CC3=CC=CC=C3)C(=O)[O-].O.O.[Ca+2]
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Chemical Name2H-Isoindole-2-butanoic acid, octahydro-γ-oxo-α-(phenylmethyl)-, calcium salt, hydrate (2:1:2), (αS,3aR,7aS)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ohnota H, et al. J Pharmacol Exp Ther. 1994 May;269(2):489-95.
2. Ohnota H, et al. Biochem Pharmacol. 1995 Jan 18;49(2):165-71.
3. Kinukawa M, et al. Br J Pharmacol. 1996 Apr;117(8):1702-6.
2. Ohnota H, et al. Biochem Pharmacol. 1995 Jan 18;49(2):165-71.
3. Kinukawa M, et al. Br J Pharmacol. 1996 Apr;117(8):1702-6.
molnova catalog
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